Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL12571

HYDROXYGUANIDINE SULPHATE
Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
N/C(=N\O)N/N=C\OS(=O)(=O)O

Basic Information

ChEMBL ID CHEMBL12571
Name HYDROXYGUANIDINE SULPHATE
Phase Preclinical
Structure Type MOL
InChI Key HADHZJGGNKXUCP-RJRFIUFISA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

198.2
MW (Da)
-1.96
ALogP
6
HBA
4
HBD
146.6
PSA (Ų)
0.14
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C2H6N4O5S
MW 198.16
Aromatic Rings 0
Heavy Atoms 12
NP-Likeness 0.40

Activity Summary

IC50 2 meas. best 4.78

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
L1210
CHEMBL386
IC50 4.78 4.78 16595.9 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
L1210 IC50 = 16595.87 nM 4.78 Concentration required for 50% inhibition of cell growth (L1210 Leukemia) 2991520

Literature References

PubMed DOI Target Context # Activities
2991520 10.1021/jm00146a022 Rous sarcoma virus 4
2991520 10.1021/jm00146a022 L1210 2

Data from ChEMBL 36 via Core Engine