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Compound Detail

CHEMBL1271925

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COc1cc2oc(-c3ccc(O)cc3)cc(=O)c2c(O)c1O[C@@H]1O[C@H](COC(C)=O)[C@@H](O)[C@H](O)[C@H]1O

Basic Information

ChEMBL ID CHEMBL1271925
Phase Preclinical
Structure Type MOL
InChI Key JIFPVGMUAPCSFJ-NZXWXYQFSA-N
1
Targets
3
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

504.4
MW (Da)
0.63
ALogP
12
HBA
5
HBD
185.3
PSA (Ų)
0.30
QED
2
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C24H24O12
MW 504.44
Aromatic Rings 3
Heavy Atoms 36
NP-Likeness 1.81

Activity Summary

EC50 3 meas. best 4.91

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
EC50 4.91 4.91 12300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET EC50 = 12300.0 nM 4.91 Antioxidant activity assessed as ABTS radical scavenging activity 20932762

Literature References

PubMed DOI Target Context # Activities
20932762 10.1016/j.bmcl.2010.09.086 NON-PROTEIN TARGET 2
20932762 10.1016/j.bmcl.2010.09.086 Radical scavenging activity 1
20932762 10.1016/j.bmcl.2010.09.086 H9c2 1

Data from ChEMBL 36 via Core Engine