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Compound Detail

CHEMBL1445768

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Cl.O=C(Oc1cccc2cccnc12)c1cccs1

Basic Information

ChEMBL ID CHEMBL1445768
Phase Preclinical
Structure Type MOL
InChI Key LYWBUZFSUSAVGV-UHFFFAOYSA-N
Parent Compound CHEMBL1621743
Active Moiety CHEMBL1621743
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

255.3
MW (Da)
3.52
ALogP
4
HBA
0
HBD
39.2
PSA (Ų)
0.52
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C14H10ClNO2S
MW 291.76
Aromatic Rings 3
Heavy Atoms 18
NP-Likeness -1.56

Activity Summary

EC50 2 meas. best 5.46

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 5.46 5.41 3460.0 2

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine