Assay Detail
Functional
CHEMBL1614320
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescent HTS Cytotoxicity/Cell viability assay (HPDE-C7K cells). (Class of assay: confirmatory) [Related pubchem assays: 430 ]
386
Total Activities
386
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 386 | 5.14 | 7.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL513000 | — | — | 1 | 7.05 |
| CHEMBL1598493 | — | — | 1 | 6.68 |
| CHEMBL3192995 | — | — | 1 | 6.62 |
| CHEMBL251785 | — | — | 1 | 6.52 |
| CHEMBL1349063 | — | — | 1 | 6.41 |
| CHEMBL578512 | — | — | 1 | 6.19 |
| CHEMBL1329237 | — | — | 1 | 5.97 |
| CHEMBL1588762 | — | — | 1 | 5.96 |
| CHEMBL16223 | — | — | 1 | 5.94 |
| CHEMBL1981770 | — | — | 1 | 5.92 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 5.87 |
| CHEMBL1582505 | — | — | 1 | 5.83 |
| CHEMBL1347618 | — | — | 1 | 5.82 |
| CHEMBL1444449 | — | — | 1 | 5.75 |
| CHEMBL1502512 | — | — | 1 | 5.68 |
| CHEMBL1566928 | — | — | 1 | 5.68 |
| CHEMBL1346587 | — | — | 1 | 5.67 |
| CHEMBL3145067 | — | — | 1 | 5.66 |
| CHEMBL1523206 | — | — | 1 | 5.66 |
| CHEMBL1532544 | — | — | 1 | 5.62 |
| CHEMBL123 | ELLIPTECINE | — | 1 | 5.62 |
| CHEMBL1383144 | — | — | 1 | 5.61 |
| CHEMBL1465527 | — | — | 1 | 5.60 |
| CHEMBL89445 | TERPYRIDINE | — | 1 | 5.59 |
| CHEMBL1430895 | — | — | 1 | 5.56 |
| CHEMBL3193792 | — | — | 1 | 5.55 |
| CHEMBL497 | CLIOQUINOL | 4.0 | 1 | 5.54 |
| CHEMBL3190220 | — | — | 1 | 5.53 |
| CHEMBL1445710 | — | — | 1 | 5.52 |
| CHEMBL1342448 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL513000 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL1598493 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL3192995 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL251785 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL1349063 | — | EC50 | = | 390.0 | nM | 6.41 |
| CHEMBL578512 | — | EC50 | = | 640.0 | nM | 6.19 |
| CHEMBL1329237 | — | EC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL1588762 | — | EC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL16223 | — | EC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL1981770 | — | EC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL290106 | BITHIONOL | EC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL1582505 | — | EC50 | = | 1490.0 | nM | 5.83 |
| CHEMBL1347618 | — | EC50 | = | 1530.0 | nM | 5.82 |
| CHEMBL1444449 | — | EC50 | = | 1770.0 | nM | 5.75 |
| CHEMBL1502512 | — | EC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL1566928 | — | EC50 | = | 2080.0 | nM | 5.68 |
| CHEMBL1346587 | — | EC50 | = | 2150.0 | nM | 5.67 |
| CHEMBL1523206 | — | EC50 | = | 2180.0 | nM | 5.66 |
| CHEMBL3145067 | — | EC50 | = | 2210.0 | nM | 5.66 |
| CHEMBL1532544 | — | EC50 | = | 2380.0 | nM | 5.62 |
| CHEMBL123 | ELLIPTECINE | EC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1383144 | — | EC50 | = | 2440.0 | nM | 5.61 |
| CHEMBL1465527 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL89445 | TERPYRIDINE | EC50 | = | 2540.0 | nM | 5.59 |
| CHEMBL1430895 | — | EC50 | = | 2730.0 | nM | 5.56 |
| CHEMBL3193792 | — | EC50 | = | 2830.0 | nM | 5.55 |
| CHEMBL497 | CLIOQUINOL | EC50 | = | 2920.0 | nM | 5.54 |
| CHEMBL3190220 | — | EC50 | = | 2940.0 | nM | 5.53 |
| CHEMBL1445710 | — | EC50 | = | 3010.0 | nM | 5.52 |
| CHEMBL1331573 | — | EC50 | = | 3060.0 | nM | 5.51 |
| CHEMBL1342448 | — | EC50 | = | 3090.0 | nM | 5.51 |
| CHEMBL1418818 | — | EC50 | = | 3170.0 | nM | 5.50 |
| CHEMBL1557648 | — | EC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL1607568 | — | EC50 | = | 3150.0 | nM | 5.50 |
| CHEMBL1200916 | THIORIDAZINE HYDROCHLORIDE | EC50 | = | 3430.0 | nM | 5.46 |
| CHEMBL1371774 | — | EC50 | = | 3470.0 | nM | 5.46 |
| CHEMBL1458840 | — | EC50 | = | 3450.0 | nM | 5.46 |
| CHEMBL1571874 | — | EC50 | = | 3540.0 | nM | 5.45 |
| CHEMBL1608535 | — | EC50 | = | 3720.0 | nM | 5.43 |
| CHEMBL1540038 | — | EC50 | = | 3680.0 | nM | 5.43 |
| CHEMBL1331809 | — | EC50 | = | 3750.0 | nM | 5.43 |
| CHEMBL1525298 | DIETHYLSTILBESTROL DIPROPIONATE | EC50 | = | 3870.0 | nM | 5.41 |
| CHEMBL1362096 | — | EC50 | = | 3890.0 | nM | 5.41 |
| CHEMBL1327738 | — | EC50 | = | 4110.0 | nM | 5.39 |
| CHEMBL261131 | DIACYLGLYCEROL KINASE INHIBITOR II | EC50 | = | 4210.0 | nM | 5.38 |
| CHEMBL1540956 | — | EC50 | = | 4170.0 | nM | 5.38 |
| CHEMBL1505922 | — | EC50 | = | 4260.0 | nM | 5.37 |
| CHEMBL1445768 | — | EC50 | = | 4380.0 | nM | 5.36 |
| CHEMBL1429929 | — | EC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL1311755 | — | EC50 | = | 4420.0 | nM | 5.36 |