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Compound Detail

CHEMBL177114

MALONIC ACID DIETHYL ESTER
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CCOC(=O)CC(=O)OCC

Basic Information

ChEMBL ID CHEMBL177114
Name MALONIC ACID DIETHYL ESTER
Phase Preclinical
Structure Type MOL
InChI Key IYXGSMUGOJNHAZ-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

160.2
MW (Da)
0.50
ALogP
4
HBA
0
HBD
52.6
PSA (Ų)
0.44
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C7H12O4
MW 160.17
Aromatic Rings 0
Heavy Atoms 11
NP-Likeness 0.14

Activity Summary

IC50 1 meas. best 5.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Alpha glucosidase
CHEMBL3833502
IC50 5.3 5.3 5000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Alpha glucosidase IC50 = 5000.0 nM 5.3 Inhibition of alpha-glucosidase (unknown origin) 31112894

Literature References

PubMed DOI Target Context # Activities
7328595 10.1021/jm00140a003 Mus musculus 2
31112894 10.1016/j.ejmech.2019.04.025 Alpha glucosidase 1

Data from ChEMBL 36 via Core Engine