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Compound Detail

CHEMBL1771752

3-CHLORO-CINNAMIC ACID
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O=C(O)/C=C/c1cccc(Cl)c1

Basic Information

ChEMBL ID CHEMBL1771752
Name 3-CHLORO-CINNAMIC ACID
Phase Preclinical
Structure Type MOL
InChI Key FFKGOJWPSXRALK-SNAWJCMRSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

182.6
MW (Da)
2.44
ALogP
1
HBA
1
HBD
37.3
PSA (Ų)
0.71
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C9H7ClO2
MW 182.61
Aromatic Rings 1
Heavy Atoms 12
NP-Likeness -0.33

Activity Summary

IC50 1 meas. best 4.86

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.86 4.86 13700.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 13700.0 nM 4.86 Antagonist activity at Gloeobacter violaceus ligand-gated ion channel expressed ... 23682762

Literature References

PubMed DOI Target Context # Activities
19368353 10.1021/jf8034385 Radish 3
23682762 10.1021/jm400374q Unchecked 2
21167710 10.1016/j.bmcl.2010.11.091 Hydroxycarboxylic acid receptor 2 1
23682762 10.1021/jm400374q No relevant target 1

Data from ChEMBL 36 via Core Engine