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Compound Detail

CHEMBL1779299

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CC(C)CCN(CCc1c[nH]c2ccccc12)CC(C)C

Basic Information

ChEMBL ID CHEMBL1779299
Phase Preclinical
Structure Type MOL
InChI Key NJVRJDGDBJWRQN-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

286.5
MW (Da)
4.71
ALogP
1
HBA
1
HBD
19.0
PSA (Ų)
0.74
QED
0
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H30N2
MW 286.46
Aromatic Rings 2
Heavy Atoms 21
NP-Likeness -0.72

Activity Summary

IC50 1 meas. best 5.96

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis B virus
CHEMBL613497
IC50 5.96 5.96 1100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Hepatitis B virus IC50 = 1100.0 nM 5.96 Antiviral activity against Hepatitis B virus infected in human HepG2(2.2.15) cel... 21524588

Literature References

PubMed DOI Target Context # Activities
21524588 10.1016/j.bmc.2011.04.004 ADMET 1
21524588 10.1016/j.bmc.2011.04.004 Unchecked 1
21524588 10.1016/j.bmc.2011.04.004 Hepatitis B virus 1

Data from ChEMBL 36 via Core Engine