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Compound Detail

CHEMBL2031684

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CC(C)(C)C(=O)SCCOP(=O)(OCCSC(=O)C(C)(C)C)OC[C@H]1O[C@@H](c2cnc3c(=O)[nH]c(N)nn23)[C@](C)(O)[C@@H]1O

Basic Information

ChEMBL ID CHEMBL2031684
Phase Preclinical
Structure Type MOL
InChI Key XMFLDCOKSOTQIU-LQIAVNJRSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

665.7
MW (Da)
2.32
ALogP
16
HBA
4
HBD
217.7
PSA (Ų)
0.19
QED
2
Ro5 Violations
12
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H40N5O10PS2
MW 665.73
Aromatic Rings 2
Heavy Atoms 43
NP-Likeness 0.32

Activity Summary

EC50 1 meas. best 5.02

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 5.02 5.02 9540.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Hepatitis C virus EC50 = 9540.0 nM 5.02 Antiviral activity against HCV genotype 1b infected in human HuH7 cells assessed... 22578461

Literature References

PubMed DOI Target Context # Activities
22578461 10.1016/j.bmcl.2012.04.065 Hepatitis C virus 1

Data from ChEMBL 36 via Core Engine