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Compound Detail

CHEMBL2042320

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Nc1nc(N)c2c(OCC(F)(F)F)cccc2n1

Basic Information

ChEMBL ID CHEMBL2042320
Phase Preclinical
Structure Type MOL
InChI Key CMIRUHXLWHGPHN-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

258.2
MW (Da)
1.74
ALogP
5
HBA
2
HBD
87.0
PSA (Ų)
0.86
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H9F3N4O
MW 258.20
Aromatic Rings 2
Heavy Atoms 18
NP-Likeness -1.20

Activity Summary

EC50 1 meas. best 8.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
dengue virus type 2
CHEMBL613966
EC50 8.1 8.1 7.9 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
22448770 10.1021/jm2015952 dengue virus type 2 1
22448770 10.1021/jm2015952 ADMET 1
22448770 10.1021/jm2015952 Unchecked 1

Data from ChEMBL 36 via Core Engine