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Compound Detail

CHEMBL206725

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N[C@@H](CCCCN(O)C=O)C(=O)O

Basic Information

ChEMBL ID CHEMBL206725
Phase Preclinical
Structure Type MOL
InChI Key YNVSSYWJQVVFPB-LURJTMIESA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

190.2
MW (Da)
-0.58
ALogP
4
HBA
3
HBD
103.9
PSA (Ų)
0.22
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C7H14N2O4
MW 190.20
Aromatic Rings 0
Heavy Atoms 13
NP-Likeness 0.97

Activity Summary

Ki 1 meas. best 4.17

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
S-ribosylhomocysteine lyase
CHEMBL5171
Ki 4.17 4.17 68000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
S-ribosylhomocysteine lyase Ki = 68000.0 nM 4.17 Inhibition of cobalt substituted Bacillus subtilis LuxS 16686542

Literature References

PubMed DOI Target Context # Activities
16686542 10.1021/jm060047g S-ribosylhomocysteine lyase 5

Data from ChEMBL 36 via Core Engine