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Compound Detail

CHEMBL2069034

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CN(C)CCCS[C@H]1CC[C@@]2(C)[C@H](CC[C@@H]3[C@@H]2CC[C@]2(C)[C@@H](C4=CC(=O)OC4)CC[C@]32O)C1

Basic Information

ChEMBL ID CHEMBL2069034
Phase Preclinical
Structure Type MOL
InChI Key GUSYJUZZKLQMPD-WRUTXJEYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

475.7
MW (Da)
5.30
ALogP
5
HBA
1
HBD
49.8
PSA (Ų)
0.42
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H45NO3S
MW 475.74
Aromatic Rings 0
Heavy Atoms 33
NP-Likeness 2.01

Activity Summary

IC50 1 meas. best 7.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 7.0 7.0 100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 100.0 nM 7.0 Displacement of [3H]ouabain binding from Na+,K+ -ATPase receptor isolated from d... -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(97)00039-5 Unchecked 1

Data from ChEMBL 36 via Core Engine