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Compound Detail

CHEMBL2087203

TERMINAMINE E
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CC(C)=C1CN([C@@H]2CC[C@@]3(C)[C@@H](CC[C@@H]4[C@@H]3CC[C@]3(C)[C@@H]([C@H](C)N(C)C)CC[C@@H]43)[C@H]2O)C1=O

Basic Information

ChEMBL ID CHEMBL2087203
Name TERMINAMINE E
Phase Preclinical
Structure Type MOL
InChI Key ZHEKCAHHEJODEA-WXWFEBHUSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

456.7
MW (Da)
5.11
ALogP
3
HBA
1
HBD
43.8
PSA (Ų)
0.47
QED
1
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C29H48N2O2
MW 456.72
Aromatic Rings 0
Heavy Atoms 33
NP-Likeness 2.21

Activity Summary

IC50 1 meas. best 7.16

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
MDA-MB-231
CHEMBL400
IC50 7.16 7.16 70.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
MDA-MB-231 IC50 = 70.0 nM 7.16 Inhibition of epithelial growth factor-induced cell migration of human MDA-MB-23... 22804108

Literature References

PubMed DOI Target Context # Activities
22804108 10.1021/np300207c MDA-MB-231 1

Data from ChEMBL 36 via Core Engine