Compound Detail

CHEMBL2107799

FLURPIRIDAZ F 18

💊 Approved Drug

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💊 Approved Drug

CC(C)(C)n1ncc(OCc2ccc(COCC[18F])cc2)c(Cl)c1=O

ChEMBL ↗ Properties Compare Identifier

Basic Information

ChEMBL ID	CHEMBL2107799
Name	FLURPIRIDAZ F 18
Phase	Approved
Structure Type	MOL
InChI Key	RMXZKEPDYBTFOS-LRFGSCOBSA-N
Parent Compound	CHEMBL494622
Active Moiety	CHEMBL494622

Known Names

BMS 747158-02 Bms-747158 BMS-747158-02 Flurpiridaz (18f) Flurpiridaz f 18 Flurpiridaz f-18 Flurpiridaz, f-18 Flyrcado

Targets

Activities

Assay Types

PK Parameters

Publications

Known Names

Indications

Mechanisms

Molecular Properties

368.8

MW (Da)

3.72

ALogP

HBA

HBD

53.4

PSA (Å²)

0.70

QED

Ro5 Violations

Rot. Bonds

Drug Information

Molecule Type	Small molecule
First Approval	2024
Availability	Prescription
Chirality	Achiral

Routes of Administration

Parenteral

USAN Year

2009

Extended Properties

Molecular Formula	C18H22ClFN2O3
MW	367.84
Aromatic Rings	2
Heavy Atoms	25
NP-Likeness	-1.08

Mechanism of Action

Mechanism	Action Type	Target	Direct	Efficacy
Diagnostic agent	-	-	✓	✓

Indications

Myocardial Perfusion Imaging Positron-Emission Tomography

Literature References

PubMed	DOI	Target Context	# Activities
23210516	10.1021/jm301453p	Nucleic Acid	3
23210516	10.1021/jm301453p	Heart	2
23210516	10.1021/jm301453p	Liver	2

Data from ChEMBL 36 via Core Engine