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Compound Detail

CHEMBL2228069

6-F-2-Et-D-DIBOA
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CCC1Oc2ccc(F)cc2N(O)C1=O

Basic Information

ChEMBL ID CHEMBL2228069
Name 6-F-2-Et-D-DIBOA
Phase Preclinical
Structure Type MOL
InChI Key GCHHILUFDJMNNE-UHFFFAOYSA-N
6
Targets
6
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

211.2
MW (Da)
1.72
ALogP
3
HBA
1
HBD
49.8
PSA (Ų)
0.72
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H10FNO3
MW 211.19
Aromatic Rings 1
Heavy Atoms 15
NP-Likeness -0.45

Activity Summary

IC50 6 meas. best 6.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Lepidium sativum
CHEMBL612381
IC50 6.0 6.0 1000.0 1
Allium cepa
CHEMBL613790
IC50 5.89 5.89 1300.0 1
Oryza sativa
CHEMBL613061
IC50 4.82 4.82 15000.0 1
Avena fatua
CHEMBL612834
IC50 4.61 4.61 24400.0 1
Echinochloa crus-galli
CHEMBL612343
IC50 4.6 4.6 25000.0 1
Triticum aestivum
CHEMBL612836
IC50 4.2 4.2 63130.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
20014762 10.1021/jf903445m Allium cepa 3
20628996 10.1002/ps.1992 Avena fatua 3
20628996 10.1002/ps.1992 Echinochloa crus-galli 3
20014762 10.1021/jf903445m Lepidium sativum 2
20628996 10.1002/ps.1992 Unchecked 2
20628996 10.1002/ps.1992 Triticum aestivum 2
20628996 10.1002/ps.1992 Oryza sativa 2
20014762 10.1021/jf903445m Lactuca sativa 1
20014762 10.1021/jf903445m Solanum lycopersicum 1

Data from ChEMBL 36 via Core Engine