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Compound Detail

CHEMBL2228074

6-Cl-2-Et-D-DIBOA
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CCC1Oc2ccc(Cl)cc2N(O)C1=O

Basic Information

ChEMBL ID CHEMBL2228074
Name 6-Cl-2-Et-D-DIBOA
Phase Preclinical
Structure Type MOL
InChI Key XQGOTDCLNUXWBR-UHFFFAOYSA-N
4
Targets
7
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

227.7
MW (Da)
2.23
ALogP
3
HBA
1
HBD
49.8
PSA (Ų)
0.75
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H10ClNO3
MW 227.65
Aromatic Rings 1
Heavy Atoms 15
NP-Likeness -0.26

Activity Summary

IC50 7 meas. best 6.4

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Lepidium sativum
CHEMBL612381
IC50 6.4 6.4 400.0 1
Allium cepa
CHEMBL613790
IC50 5.8 5.8 1600.0 1
Solanum lycopersicum
CHEMBL613317
IC50 5.64 5.64 2300.0 1
Oryza sativa
CHEMBL613061
IC50 4.25 4.25 56000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
20014762 10.1021/jf903445m Allium cepa 3
20014762 10.1021/jf903445m Lepidium sativum 3
20628996 10.1002/ps.1992 Avena fatua 3
20628996 10.1002/ps.1992 Echinochloa crus-galli 3
20014762 10.1021/jf903445m Solanum lycopersicum 2
20628996 10.1002/ps.1992 Unchecked 2
20628996 10.1002/ps.1992 Triticum aestivum 2
20628996 10.1002/ps.1992 Oryza sativa 2
20014762 10.1021/jf903445m Lactuca sativa 1

Data from ChEMBL 36 via Core Engine