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Compound Detail

CHEMBL2348117

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O=C(Nc1ccccc1[N+](=O)[O-])c1cc(Cl)ccc1O

Basic Information

ChEMBL ID CHEMBL2348117
Phase Preclinical
Structure Type MOL
InChI Key ALSFHFRMXBCGJT-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

292.7
MW (Da)
3.21
ALogP
4
HBA
2
HBD
92.5
PSA (Ų)
0.67
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H9ClN2O4
MW 292.68
Aromatic Rings 2
Heavy Atoms 20
NP-Likeness -1.73

Activity Summary

IC50 2 meas. best 5.23

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.23 5.02 5850.0 2

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 5850.0 nM 5.23 Inhibition of envelope protein in Zika virus 33689873
Unchecked IC50 = 15590.0 nM 4.81 Inhibition of NS-1in Zika virus 33689873

Literature References

PubMed DOI Target Context # Activities
33689873 10.1016/j.bmcl.2021.127906 Unchecked 2
33689873 10.1016/j.bmcl.2021.127906 ADMET 2
23453073 10.1016/j.bmcl.2013.01.101 Molecular identity unknown 1
23453073 10.1016/j.bmcl.2013.01.101 Frizzled-1 1
33689873 10.1016/j.bmcl.2021.127906 No relevant target 1

Data from ChEMBL 36 via Core Engine