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Compound Detail

CHEMBL265719

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Nc1cc(OC[C@@H](CO)OCP(=O)(O)O)nc(N)n1

Basic Information

ChEMBL ID CHEMBL265719
Phase Preclinical
Structure Type MOL
InChI Key SDORNFBUOMQVCA-RXMQYKEDSA-N
2
Targets
7
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

294.2
MW (Da)
-1.47
ALogP
8
HBA
5
HBD
174.0
PSA (Ų)
0.37
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H15N4O6P
MW 294.20
Aromatic Rings 1
Heavy Atoms 19
NP-Likeness 0.31

Activity Summary

EC50 7 meas. best 5.09

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
EC50 5.09 4.965 8200.0 4
Simian virus 40
CHEMBL613051
EC50 4.14 4.14 72800.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
17420214 10.1128/aac.01422-06 Unchecked 7
17420214 10.1128/aac.01422-06 NON-PROTEIN TARGET 4
17420214 10.1128/aac.01422-06 Simian virus 40 3
17420214 10.1128/aac.01422-06 ADMET 2

Data from ChEMBL 36 via Core Engine