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Compound Detail

CHEMBL26801

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Nc1ncnc2c1nnn2C1CC(CO)C(O)C1O

Basic Information

ChEMBL ID CHEMBL26801
Phase Preclinical
Structure Type MOL
InChI Key XKNNLGAIRDUJOQ-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

266.3
MW (Da)
-1.92
ALogP
9
HBA
4
HBD
143.2
PSA (Ų)
0.49
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C10H14N6O3
MW 266.26
Aromatic Rings 2
Heavy Atoms 19
NP-Likeness 0.33

Activity Summary

Ki 1 meas. best 4.66

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Adenosylhomocysteinase
CHEMBL2664
Ki 4.66 4.66 22000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Adenosylhomocysteinase Ki = 22000.0 nM 4.66 Binding affinity against S-adenosyl-homocysteine hydrolase 3981539

Literature References

PubMed DOI Target Context # Activities
6481772 10.1021/jm00376a025 Mus musculus 10
3981539 10.1021/jm00382a015 Adenosylhomocysteinase 2
3981539 10.1021/jm00382a015 L cells 2
1433208 10.1021/jm00100a003 P388 1
3981539 10.1021/jm00382a015 L929 1

Data from ChEMBL 36 via Core Engine