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Compound Detail

CHEMBL275722

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COC[C@H]1OC(=O)c2coc3c2[C@@]1(C)C1=C(C3=O)[C@@H]2CC=C(OC(C)=O)[C@@]2(C)C[C@H]1OC(C)=O

Basic Information

ChEMBL ID CHEMBL275722
Phase Preclinical
Structure Type MOL
InChI Key WBRDXASLVDYYMQ-JDQULTIISA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

470.5
MW (Da)
3.02
ALogP
9
HBA
0
HBD
118.3
PSA (Ų)
0.48
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H26O9
MW 470.47
Aromatic Rings 1
Heavy Atoms 34
NP-Likeness 2.43

Activity Summary

IC50 1 meas. best 7.23

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 7.23 7.23 59.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 59.0 nM 7.23 In vitro inhibitory activity against Phosphatidylinositol 3-Kinase 8676346

Literature References

PubMed DOI Target Context # Activities
8676346 10.1021/jm950619p Unchecked 1

Data from ChEMBL 36 via Core Engine