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Compound Detail

CHEMBL279597

ALANINE
🧪 Phase III
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🧪 Phase III
C[C@H](N)C(=O)O

Basic Information

ChEMBL ID CHEMBL279597
Name ALANINE
Phase Phase III
Structure Type MOL
InChI Key QNAYBMKLOCPYGJ-REOHCLBHSA-N

Known Names

(2s)-2-aminopropanoic acid Alanina Alanine E639 L-2-aminopropanoic acid L-alanine NSC-206315
1
Targets
3
Activities
2
Assay Types
4
PK Parameters
20
Publications
7
Known Names
7
Indications

Molecular Properties

89.1
MW (Da)
-0.58
ALogP
2
HBA
2
HBD
63.3
PSA (Ų)
0.45
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Chirality Single Enantiomer

Flags

Natural Product
USAN Year 1979

Extended Properties

Molecular Formula C3H7NO2
MW 89.09
Aromatic Rings 0
Heavy Atoms 6
NP-Likeness 0.38

Indications

Coronary Disease Asthma Fructose Intolerance Alzheimer Disease Cognitive Dysfunction Glioma Severe Acute Respiratory Syndrome

Activity Summary

IC50 2 meas. best 4.11
Ki 1 meas.

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.11 4.11 78000.0 1

Pharmacokinetic Data

Parameter Value Units Species
KA 54.0 uM -
KA 150.0 uM -
KA 66.0 uM -
T1/2 1.292 hr Canis lupus familiaris

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 78000.0 nM 4.11 Inhibition of binding of [3H]strychnine to N-methyl-D-aspartate glutamate recept... 2549245

Literature References

PubMed DOI Target Context # Activities
18794383 10.1128/aac.01648-07 Saccharomyces cerevisiae 7
37731697 10.1039/d3md00274h Jurkat E6.1 6
23324083 10.1021/jm301407k No relevant target 6
23324083 10.1021/jm301407k Lipopolysaccharide (LPS) 5
23324083 10.1021/jm301407k RAW264.7 5
23324083 10.1021/jm301407k ADMET 4
23324083 10.1021/jm301407k Staphylococcus aureus 3
23324083 10.1021/jm301407k Escherichia coli 3
- 10.6019/CHEMBL4808148 Histone deacetylase 6 2
37468498 10.1038/s41467-023-40064-9 Alpha-1A adrenergic receptor 2
32182061 10.1021/acs.jmedchem.9b01877 Alanine racemase, biosynthetic 2
7252987 10.1021/jm00138a026 Canis familiaris 2
37468498 10.1038/s41467-023-40064-9 Thromboxane A2 receptor 2
- 10.6019/CHEMBL4495565 SARS-CoV-2 2
37468498 10.1038/s41467-023-40064-9 Prostaglandin G/H synthase 1 2
21955456 10.1016/j.bmc.2011.08.058 Proton-coupled amino acid transporter 1 2
37468498 10.1038/s41467-023-40064-9 Muscarinic acetylcholine receptor M1 2
12729634 10.1016/s0960-894x(03)00280-4 Unchecked 1
3656360 10.1021/jm00393a031 Unchecked 1
3079831 10.1021/jm00151a024 Alanine racemase, biosynthetic 1

Data from ChEMBL 36 via Core Engine