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Compound Detail

CHEMBL287845

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Nc1nc(=O)n(COC(CO)CO)cc1F

Basic Information

ChEMBL ID CHEMBL287845
Phase Preclinical
Structure Type MOL
InChI Key IWVFFRUDPUZDMN-UHFFFAOYSA-N
1
Targets
2
Activities
2
Assay Types
0
PK Parameters
8
Publications
0
Known Names

Molecular Properties

233.2
MW (Da)
-1.71
ALogP
7
HBA
3
HBD
110.6
PSA (Ų)
0.56
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H12FN3O4
MW 233.20
Aromatic Rings 1
Heavy Atoms 16
NP-Likeness 0.03

Activity Summary

EC50 1 meas.
IC50 1 meas. best 4.85

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Cytomegalovirus
CHEMBL613134
IC50 4.85 4.85 14000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Cytomegalovirus IC50 = 14000.0 nM 4.85 Inhibition of growth of human cytomegalovirus (HCMV) was determined by plaque re... 2826784

Literature References

PubMed DOI Target Context # Activities
16759112 10.1021/jm060102l Hepatitis B virus 3
16759112 10.1021/jm060102l Duck hepatitis B virus 2
2826784 10.1021/jm00396a021 Cytomegalovirus 1
2826784 10.1021/jm00396a021 Human gammaherpesvirus 4 1
3871860 10.1021/jm00381a015 Vero 1
16759112 10.1021/jm060102l HepG2 1
16759112 10.1021/jm060102l Vero 1
16759112 10.1021/jm060102l Hepatitis C virus 1

Data from ChEMBL 36 via Core Engine