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Compound Detail

CHEMBL3098861

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COc1cc(C[C@@H]2COC(=O)[C@@]2(Cc2ccc(O)c(OC)c2)O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)ccc1O

Basic Information

ChEMBL ID CHEMBL3098861
Phase Preclinical
Structure Type MOL
InChI Key YAVQULWQXQRTKS-QDYGYTTASA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

536.5
MW (Da)
-0.37
ALogP
12
HBA
6
HBD
184.6
PSA (Ų)
0.23
QED
3
Ro5 Violations
9
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C26H32O12
MW 536.53
Aromatic Rings 2
Heavy Atoms 38
NP-Likeness 1.53

Activity Summary

IC50 1 meas. best 4.38

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.38 4.38 41200.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 41200.0 nM 4.38 Inhibition of Streptococcus mutans OMZ65 recombinant sortase A delta-40 mutant u... 24360605

Literature References

PubMed DOI Target Context # Activities
24360605 10.1016/j.bmcl.2013.12.006 Unchecked 1

Data from ChEMBL 36 via Core Engine