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Compound Detail

CHEMBL3109438

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COc1c(O)cc(-c2oc3cc(O)cc(O)c3c(=O)c2O[C@@H]2O[C@@H](C)[C@H](O)[C@@H](O)[C@H]2O)cc1O

Basic Information

ChEMBL ID CHEMBL3109438
Phase Preclinical
Structure Type MOL
InChI Key NAQNISJXKDSYJD-DHWIRCOFSA-N
1
Targets
3
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

478.4
MW (Da)
0.50
ALogP
12
HBA
7
HBD
199.5
PSA (Ų)
0.27
QED
2
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C22H22O12
MW 478.41
Aromatic Rings 3
Heavy Atoms 34
NP-Likeness 2.14

Activity Summary

IC50 3 meas. best 5.72

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
No relevant target
CHEMBL2362975
IC50 5.72 5.72 1900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
No relevant target IC50 = 1900.0 nM 5.72 Antioxidant activity assessed as DPPH radical scavenging activity measured after... 29300477

Literature References

PubMed DOI Target Context # Activities
24521209 10.1021/np400717m Arginase 1
29300477 10.1021/acs.jnatprod.7b00564 Tyrosinase 1
29300477 10.1021/acs.jnatprod.7b00564 No relevant target 1

Data from ChEMBL 36 via Core Engine