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Assay Detail

CHEMBL4136835

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Functional
Antioxidant activity assessed as DPPH radical scavenging activity measured after 30 mins incubation under dark condition
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Publication

Isolation of Flavonoids and Flavonoid Glycosides from Myrsine africana and Their Inhibitory Activities against Mushroom Tyrosinase.
Kishore N, Twilley D, Blom van Staden A, Verma P, Singh B, Cardinali G, Kovacs D, Picardo M, Kumar V, Lall N.
J Nat Prod (2018) 81 : 49 -56
PubMed 29300477 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 13 5.51 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3109438 1 5.72
CHEMBL522983 1 5.70
CHEMBL4176025 1 5.66
CHEMBL82242 QUERCITRIN 1 5.66
CHEMBL226335 RUTIN 3.0 1 5.64
CHEMBL4163708 1 5.52
CHEMBL50 QUERCETIN 3.0 1 5.50
CHEMBL4164304 1 5.50
CHEMBL4172192 1 5.47
CHEMBL4167746 1 5.46
CHEMBL4168843 1 5.41
CHEMBL164 MYRICETIN 1 5.38
CHEMBL196 ASCORBIC ACID 4.0 1 4.95

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3109438 IC50 = 1900.0 nM 5.72
CHEMBL522983 IC50 = 2000.0 nM 5.70
CHEMBL4176025 IC50 = 2200.0 nM 5.66
CHEMBL82242 QUERCITRIN IC50 = 2200.0 nM 5.66
CHEMBL226335 RUTIN IC50 = 2300.0 nM 5.64
CHEMBL4163708 IC50 = 3000.0 nM 5.52
CHEMBL50 QUERCETIN IC50 = 3200.0 nM 5.50
CHEMBL4164304 IC50 = 3200.0 nM 5.50
CHEMBL4172192 IC50 = 3400.0 nM 5.47
CHEMBL4167746 IC50 = 3500.0 nM 5.46
CHEMBL4168843 IC50 = 3900.0 nM 5.41
CHEMBL164 MYRICETIN IC50 = 4200.0 nM 5.38
CHEMBL196 ASCORBIC ACID IC50 = 11200.0 nM 4.95