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Compound Detail

CHEMBL3143179

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O=c1nc2oc(CCCCCCCCCF)cc2cn1[C@H]1C[C@H](O)[C@@H](CO)O1

Basic Information

ChEMBL ID CHEMBL3143179
Phase Preclinical
Structure Type MOL
InChI Key BDHNAZQUWYSHJE-RCCFBDPRSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
7
Publications
0
Known Names

Molecular Properties

396.5
MW (Da)
2.87
ALogP
7
HBA
2
HBD
97.7
PSA (Ų)
0.57
QED
0
Ro5 Violations
11
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C20H29FN2O5
MW 396.46
Aromatic Rings 2
Heavy Atoms 28
NP-Likeness 0.66

Activity Summary

EC50 2 meas. best 7.85

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 3
CHEMBL613132
EC50 7.85 7.755 14.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
10866384 10.1016/s0960-894x(00)00193-1 Human alphaherpesvirus 3 4
10866384 10.1016/s0960-894x(00)00193-1 NON-PROTEIN TARGET 1
10866384 10.1016/s0960-894x(00)00193-1 HEL 1
10866384 10.1016/s0960-894x(00)00193-1 Human alphaherpesvirus 1 1
10866384 10.1016/s0960-894x(00)00193-1 Human alphaherpesvirus 2 1
10866384 10.1016/s0960-894x(00)00193-1 Cytomegalovirus 1
10866384 10.1016/s0960-894x(00)00193-1 Human immunodeficiency virus 1 1

Data from ChEMBL 36 via Core Engine