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Compound Detail

CHEMBL330156

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Cc1cc(CCCOc2c(C)cc(-c3cccc([N+](=O)[O-])c3)cc2C)on1

Basic Information

ChEMBL ID CHEMBL330156
Phase Preclinical
Structure Type MOL
InChI Key ZURRCODHMVJJKP-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

366.4
MW (Da)
5.19
ALogP
5
HBA
0
HBD
78.4
PSA (Ų)
0.33
QED
1
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H22N2O4
MW 366.42
Aromatic Rings 3
Heavy Atoms 27
NP-Likeness -1.21

Activity Summary

IC50 2 meas. best 6.46

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
rhinovirus B5
CHEMBL612467
IC50 6.46 6.46 350.0 1
Unchecked
CHEMBL612545
IC50 6.46 6.46 350.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 350.0 nM 6.46 Antiviral activity against Human rhinovirus B3 31226653
rhinovirus B5 IC50 = 350.0 nM 6.46 Antiviral activity against Human rhinovirus B5 31226653

Literature References

PubMed DOI Target Context # Activities
7629816 10.1021/jm00014a029 Human rhinovirus sp. 1
17665898 10.1021/jm0704806 rhinovirus A2 1
17665898 10.1021/jm0704806 Unchecked 1
17665898 10.1021/jm0704806 HeLa 1
31226653 10.1016/j.ejmech.2019.06.008 Unchecked 1
31226653 10.1016/j.ejmech.2019.06.008 rhinovirus B5 1

Data from ChEMBL 36 via Core Engine