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Compound Detail

CHEMBL331373

HADACIDIN
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O=CN(O)CC(=O)O

Basic Information

ChEMBL ID CHEMBL331373
Name HADACIDIN
Phase Preclinical
Structure Type MOL
InChI Key URJHVPKUWOUENU-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

119.1
MW (Da)
-1.08
ALogP
3
HBA
2
HBD
77.8
PSA (Ų)
0.28
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C3H5NO4
MW 119.08
Aromatic Rings 0
Heavy Atoms 8
NP-Likeness 0.53

Activity Summary

IC50 1 meas. best 5.46

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Adenylosuccinate synthetase isozyme 2
CHEMBL4875
IC50 5.46 5.46 3500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Adenylosuccinate synthetase isozyme 2 IC50 = 3500.0 nM 5.46 Inhibitory concentration against Adenylosuccinate synthetase 15214773

Literature References

PubMed DOI Target Context # Activities
21129960 10.1016/j.bmcl.2010.10.088 Unchecked 3
18834112 10.1021/jm800656v Amine oxidase [flavin-containing] B 2
15214773 10.1021/jm040031v Adenylosuccinate synthetase isozyme 2 1

Data from ChEMBL 36 via Core Engine