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Compound Detail

CHEMBL336343

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CCCC[C@H]1C(=O)O[C@@H]2O[C@@]3(C)CCC4[C@H](C)CC[C@@H]1[C@]42OO3

Basic Information

ChEMBL ID CHEMBL336343
Phase Preclinical
Structure Type MOL
InChI Key UYVNDCPGEVTENG-KYVWFIJHSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

324.4
MW (Da)
3.57
ALogP
5
HBA
0
HBD
54.0
PSA (Ų)
0.59
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C18H28O5
MW 324.42
Aromatic Rings 0
Heavy Atoms 23
NP-Likeness 3.38

Activity Summary

IC50 1 meas. best 4.91

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Leishmania donovani
CHEMBL367
IC50 4.91 4.91 12300.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Leishmania donovani IC50 = 12300.0 nM 4.91 Antileishmanial activity of compound against leishmania donovani was determined ... 13678403

Literature References

PubMed DOI Target Context # Activities
13678403 10.1021/jm030181q Leishmania donovani 1

Data from ChEMBL 36 via Core Engine