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Compound Detail

CHEMBL3392932

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CCC[C@@H]1C[C@@H](C(=O)N[C@H]([C@@H]2O[C@H](SC)[C@H](O)[C@@H](O)[C@H]2O)[C@@H](C)O)N(C)C1

Basic Information

ChEMBL ID CHEMBL3392932
Phase Preclinical
Structure Type MOL
InChI Key OJMMVQQUTAEWLP-UKGOLDLVSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

406.6
MW (Da)
-0.86
ALogP
8
HBA
5
HBD
122.5
PSA (Ų)
0.37
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C18H34N2O6S
MW 406.55
Aromatic Rings 0
Heavy Atoms 27
NP-Likeness 0.64

Activity Summary

IC50 1 meas. best 5.15

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Plasmodium falciparum
CHEMBL364
IC50 5.15 5.15 7080.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Plasmodium falciparum IC50 = 7080.0 nM 5.15 DNDI: Malaria in Vitro, 72 hour -

Literature References

PubMed DOI Target Context # Activities
- 10.6019/CHEMBL3392926 NON-PROTEIN TARGET 2
- 10.6019/CHEMBL3392926 Leishmania donovani 2
- 10.6019/CHEMBL3392926 Trypanosoma cruzi 1
- 10.6019/CHEMBL3392926 Plasmodium falciparum 1
- 10.6019/CHEMBL3392926 Trypanosoma brucei rhodesiense 1

Data from ChEMBL 36 via Core Engine