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Compound Detail

CHEMBL341824

PTEROIC ACID
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Nc1nc(O)c2nc(CNc3ccc(C(=O)O)cc3)cnc2n1

Basic Information

ChEMBL ID CHEMBL341824
Name PTEROIC ACID
Phase Preclinical
Structure Type MOL
InChI Key JOAQINSXLLMRCV-UHFFFAOYSA-N
1
Targets
5
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

312.3
MW (Da)
1.02
ALogP
8
HBA
4
HBD
147.1
PSA (Ų)
0.55
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C14H12N6O3
MW 312.29
Aromatic Rings 3
Heavy Atoms 23
NP-Likeness -0.73

Activity Summary

IC50 5 meas. best 4.8

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.8 4.8 16000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 16000.0 nM 4.8 Inhibitory activity against CDK4 using recombinant human cyclin D2-CDK4 complex ... 11741479

Literature References

PubMed DOI Target Context # Activities
11741479 10.1021/jm0103256 Unchecked 1
11754581 10.1021/jm010186s Ricin 1
11754581 10.1021/jm010186s Unchecked 1
21641093 10.1016/j.ejmech.2011.05.025 Ricin 1
23214944 10.1021/jm3016393 Ricin 1
321779 10.1021/jm00213a023 Enterococcus faecalis 1

Data from ChEMBL 36 via Core Engine