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Compound Detail

CHEMBL344384

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C[C@@H]([C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](N(C)C)CC[C@]4(C)[C@H]3CC[C@]12C)N(C)C

Basic Information

ChEMBL ID CHEMBL344384
Phase Preclinical
Structure Type MOL
InChI Key YTNIUPZRMQLHNV-XSIUSZODSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

372.6
MW (Da)
5.45
ALogP
2
HBA
0
HBD
6.5
PSA (Ų)
0.61
QED
1
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C25H44N2
MW 372.64
Aromatic Rings 0
Heavy Atoms 27
NP-Likeness 2.32

Activity Summary

IC50 1 meas. best 4.4

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Acetylcholinesterase
CHEMBL220
IC50 4.4 4.4 39810.7 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Acetylcholinesterase IC50 = 39810.72 nM 4.4 Compound was tested for the in silico inhibition of acetylcholinesterase 14643329

Literature References

PubMed DOI Target Context # Activities
14643329 10.1016/j.bmcl.2003.09.034 Acetylcholinesterase 1

Data from ChEMBL 36 via Core Engine