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Compound Detail

CHEMBL350934

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Nc1nc(O)c2ncn(C3CC(O)C(OCP(=O)(O)O)C3)c2n1

Basic Information

ChEMBL ID CHEMBL350934
Phase Preclinical
Structure Type MOL
InChI Key BCLMGFJGYYTZMW-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

345.2
MW (Da)
-0.67
ALogP
9
HBA
5
HBD
176.8
PSA (Ų)
0.45
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H16N5O6P
MW 345.25
Aromatic Rings 2
Heavy Atoms 23
NP-Likeness 0.52

Activity Summary

IC50 1 meas. best 5.62

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HEp-2
CHEMBL614735
IC50 5.62 5.62 2400.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HEp-2 IC50 = 2400.0 nM 5.62 Cytotoxicity to human epidermoid carcinoma cells (HEP-2) 8145223

Literature References

PubMed DOI Target Context # Activities
8145223 10.1021/jm00032a006 HEp-2 1

Data from ChEMBL 36 via Core Engine