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Compound Detail

CHEMBL362351

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O=c1ccn([C@@H]2O[C@H](CO)C(O)[C@@H]2OC2Sc3ccccc3S2)c(=O)[nH]1

Basic Information

ChEMBL ID CHEMBL362351
Phase Preclinical
Structure Type MOL
InChI Key IAAUCXKZVFNSMT-NCKWGAROSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

396.4
MW (Da)
0.35
ALogP
9
HBA
3
HBD
113.8
PSA (Ų)
0.68
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H16N2O6S2
MW 396.45
Aromatic Rings 2
Heavy Atoms 26
NP-Likeness 0.86

Activity Summary

EC50 1 meas. best 4.25

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
ADMET
CHEMBL612558
EC50 4.25 4.25 56700.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
ADMET EC50 = 56700.0 nM 4.25 Anti BVDV activity in MDBK (Madin-darby bovine kidney) cells 15456271

Literature References

PubMed DOI Target Context # Activities
15456271 10.1021/jm049677d ADMET 4

Data from ChEMBL 36 via Core Engine