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Compound Detail

CHEMBL364765

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CC(=O)OC[C@H]1S[C@@H](n2nc(C)c(=S)[nH]c2=O)C[C@@H]1OC(C)=O

Basic Information

ChEMBL ID CHEMBL364765
Phase Preclinical
Structure Type MOL
InChI Key CHJHGFGTYYTUMH-HBNTYKKESA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

359.4
MW (Da)
1.11
ALogP
9
HBA
1
HBD
103.3
PSA (Ų)
0.63
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H17N3O5S2
MW 359.43
Aromatic Rings 1
Heavy Atoms 23
NP-Likeness 0.04

Activity Summary

IC50 2 meas. best 5.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 2
CHEMBL370
IC50 5.1 5.1 8000.0 1
Human alphaherpesvirus 1
CHEMBL377
IC50 5.1 5.1 8000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
15481985 10.1021/jm049806q HEL 6
15481985 10.1021/jm049806q E6SM 5
15481985 10.1021/jm049806q ADMET 2
19112024 10.1016/j.bmc.2008.11.075 Human alphaherpesvirus 1 1
19112024 10.1016/j.bmc.2008.11.075 Human alphaherpesvirus 2 1

Data from ChEMBL 36 via Core Engine