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Compound Detail

CHEMBL374628

HYDROXYHOPANONE
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CC(C)(O)[C@H]1CC[C@@]2(C)C1CC[C@]1(C)[C@@H]2CC[C@@H]2[C@@]3(C)CCC(=O)C(C)(C)[C@@H]3CC[C@]21C

Basic Information

ChEMBL ID CHEMBL374628
Name HYDROXYHOPANONE
Phase Preclinical
Structure Type MOL
InChI Key NVNUNRUPWXZKAL-RVUONTCYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
7
Publications
0
Known Names

Molecular Properties

442.7
MW (Da)
7.43
ALogP
2
HBA
1
HBD
37.3
PSA (Ų)
0.46
QED
1
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C30H50O2
MW 442.73
Aromatic Rings 0
Heavy Atoms 32
NP-Likeness 2.51

Activity Summary

IC50 1 meas. best 4.11

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
COLO 205
CHEMBL614561
IC50 4.11 4.11 77100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
COLO 205 IC50 = 77100.0 nM 4.11 Cytotoxicity against human COLON205 cells after 48 hrs by MTT assay 17346076

Literature References

PubMed DOI Target Context # Activities
17346076 10.1021/np060631s ADMET 4
17346076 10.1021/np060631s KB 1
17346076 10.1021/np060631s K562 1
17346076 10.1021/np060631s MCF7 1
17346076 10.1021/np060631s COLO 205 1
2828553 10.1021/np50052a022 Human alphaherpesvirus 1 1
2828553 10.1021/np50052a022 Human alphaherpesvirus 2 1

Data from ChEMBL 36 via Core Engine