Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL3780638

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
COc1ccc(C(=O)NNc2c(F)cccc2F)cc1

Basic Information

ChEMBL ID CHEMBL3780638
Phase Preclinical
Structure Type MOL
InChI Key MEYNYWUBEWURPQ-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

278.3
MW (Da)
2.73
ALogP
3
HBA
2
HBD
50.4
PSA (Ų)
0.85
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C14H12F2N2O2
MW 278.26
Aromatic Rings 2
Heavy Atoms 20
NP-Likeness -1.50

Activity Summary

EC50 1 meas. best 4.13

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Enterovirus A71
CHEMBL612436
EC50 4.13 4.13 74030.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Enterovirus A71 EC50 = 74030.0 nM 4.13 Antiviral activity against Human enterovirus 71 infected in monkey African green... 26885567

Literature References

Data from ChEMBL 36 via Core Engine