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Compound Detail

CHEMBL3792660

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Cc1cccc(NC(=O)C2CSc3c(C4CC4)c(Cc4cccc5ccccc45)cc(=O)n32)c1

Basic Information

ChEMBL ID CHEMBL3792660
Phase Preclinical
Structure Type MOL
InChI Key LMSMOXORTBNOOI-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

466.6
MW (Da)
6.06
ALogP
4
HBA
1
HBD
51.1
PSA (Ų)
0.39
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C29H26N2O2S
MW 466.61
Aromatic Rings 4
Heavy Atoms 34
NP-Likeness -0.75

Activity Summary

EC50 1 meas. best 6.99

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Chlamydia trachomatis
CHEMBL614606
EC50 6.99 6.99 102.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Chlamydia trachomatis EC50 = 102.0 nM 6.99 Antimicrobial activity against Chlamydia trachomatis serovar LGV-L2 infected in ... 26849778

Literature References

PubMed DOI Target Context # Activities
26849778 10.1021/acs.jmedchem.5b01759 Chlamydia trachomatis 3
26849778 10.1021/acs.jmedchem.5b01759 HeLa 2

Data from ChEMBL 36 via Core Engine