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Compound Detail

CHEMBL3810410

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Fc1ccc(-c2nc3cc4cccnc4cc3[nH]2)c(F)c1

Basic Information

ChEMBL ID CHEMBL3810410
Phase Preclinical
Structure Type MOL
InChI Key JXLNRWQHYFVPLR-UHFFFAOYSA-N
2
Targets
3
Activities
1
Assay Types
0
PK Parameters
9
Publications
0
Known Names

Molecular Properties

281.3
MW (Da)
4.06
ALogP
2
HBA
1
HBD
41.6
PSA (Ų)
0.57
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H9F2N3
MW 281.26
Aromatic Rings 4
Heavy Atoms 21
NP-Likeness -1.45

Activity Summary

EC50 3 meas. best 5.22

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
EC50 5.22 5.11 6000.0 2
Coxsackievirus B2
CHEMBL613202
EC50 4.46 4.46 35000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
27161176 10.1016/j.ejmech.2016.03.080 ADMET 3
27161176 10.1016/j.ejmech.2016.03.080 NON-PROTEIN TARGET 2
27161176 10.1016/j.ejmech.2016.03.080 Unchecked 1
27161176 10.1016/j.ejmech.2016.03.080 Yellow fever virus 1
27161176 10.1016/j.ejmech.2016.03.080 Coxsackievirus B2 1
27161176 10.1016/j.ejmech.2016.03.080 Poliovirus 1 1
27161176 10.1016/j.ejmech.2016.03.080 Respiratory syncytial virus 1
27161176 10.1016/j.ejmech.2016.03.080 Vesicular stomatitis virus 1
27161176 10.1016/j.ejmech.2016.03.080 Vaccinia virus 1

Data from ChEMBL 36 via Core Engine