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Compound Detail

CHEMBL382689

ACETAMIDODIDEOXYNOJIRIMYCIN
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CC(=O)N[C@H]1CN[C@H](CO)[C@@H](O)[C@@H]1O

Basic Information

ChEMBL ID CHEMBL382689
Name ACETAMIDODIDEOXYNOJIRIMYCIN
Phase Preclinical
Structure Type MOL
InChI Key GBRAQQUMMCVTAV-LXGUWJNJSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

204.2
MW (Da)
-2.82
ALogP
5
HBA
5
HBD
101.8
PSA (Ų)
0.33
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H16N2O4
MW 204.23
Aromatic Rings 0
Heavy Atoms 14
NP-Likeness 1.46

Activity Summary

Ki 2 meas. best 6.16

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Ki 6.16 6.16 700.0 1
Putative beta-hexosaminidase
CHEMBL4534
Ki 4.1 4.1 80000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
23363020 10.1021/jm301557k Unchecked 2
16481162 10.1016/j.bmcl.2006.01.095 Putative beta-hexosaminidase 1

Data from ChEMBL 36 via Core Engine