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Compound Detail

CHEMBL3896035

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CCCCCCCCNC(=O)c1coc([C@@H]2CCCN2Cc2cc(F)ccc2CCC(=O)NS(=O)(=O)C(F)(F)F)n1

Basic Information

ChEMBL ID CHEMBL3896035
Phase Preclinical
Structure Type MOL
InChI Key BFFVYRGBDKURRE-QHCPKHFHSA-N
7
Targets
7
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

604.7
MW (Da)
5.14
ALogP
7
HBA
2
HBD
121.6
PSA (Ų)
0.21
QED
2
Ro5 Violations
15
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C27H36F4N4O5S
MW 604.67
Aromatic Rings 2
Heavy Atoms 41
NP-Likeness -0.82

Activity Summary

EC50 7 meas. best 7.75

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Prostaglandin D2 receptor
CHEMBL4427
EC50 7.75 7.75 18.0 1
Prostaglandin E2 receptor EP4 subtype
CHEMBL1836
EC50 7.72 7.72 19.0 1
Prostaglandin E2 receptor EP1 subtype
CHEMBL1811
EC50 7.7 7.7 20.0 1
Prostaglandin E2 receptor EP3 subtype
CHEMBL3710
EC50 6.96 6.96 110.0 1
Prostaglandin F2-alpha receptor
CHEMBL1987
EC50 6.57 6.57 270.0 1
Prostacyclin receptor
CHEMBL1995
EC50 6.54 6.54 290.0 1
Prostaglandin E2 receptor EP2 subtype
CHEMBL1881
EC50 5.6 5.6 2500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine