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Compound Detail

CHEMBL401671

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COCCc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

Basic Information

ChEMBL ID CHEMBL401671
Phase Preclinical
Structure Type MOL
InChI Key RTBVMVGMDMZLPS-UORFTKCHSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
6
Publications
0
Known Names

Molecular Properties

310.3
MW (Da)
-1.37
ALogP
9
HBA
3
HBD
122.8
PSA (Ų)
0.62
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H18N4O5
MW 310.31
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness 0.96

Activity Summary

EC50 1 meas. best 4.4

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 4.4 4.4 40000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Hepatitis C virus EC50 = 40000.0 nM 4.4 Antiviral activity against HCV 1b Con1 replicon in Huh7 cells 17997319

Literature References

Data from ChEMBL 36 via Core Engine