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Compound Detail

CHEMBL4070591

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C1=C(CCc2ccccc2)COc2ccccc21

Basic Information

ChEMBL ID CHEMBL4070591
Phase Preclinical
Structure Type MOL
InChI Key JDCYRLXBMQISAR-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

236.3
MW (Da)
4.10
ALogP
1
HBA
0
HBD
9.2
PSA (Ų)
0.78
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C17H16O
MW 236.31
Aromatic Rings 2
Heavy Atoms 18
NP-Likeness 0.66

Activity Summary

IC50 1 meas. best 6.32

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
rhinovirus A1B
CHEMBL613713
IC50 6.32 6.32 480.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
rhinovirus A1B IC50 = 480.0 nM 6.32 Antiviral activity against HRV 1B infected in human HeLa cells after 72 hrs by p... 28242170

Literature References

PubMed DOI Target Context # Activities
28242170 10.1016/j.bmc.2017.02.012 rhinovirus B14 3
28242170 10.1016/j.bmc.2017.02.012 HeLa 2
28242170 10.1016/j.bmc.2017.02.012 rhinovirus A1B 2
28242170 10.1016/j.bmc.2017.02.012 Unchecked 1

Data from ChEMBL 36 via Core Engine