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Compound Detail

CHEMBL4092514

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NCCCc1ccc(-c2ccc(-c3ccc(-c4cccs4)s3)s2)s1

Basic Information

ChEMBL ID CHEMBL4092514
Phase Preclinical
Structure Type MOL
InChI Key ZUOOWNNRXJMASV-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

387.6
MW (Da)
6.82
ALogP
5
HBA
1
HBD
26.0
PSA (Ų)
0.39
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H17NS4
MW 387.62
Aromatic Rings 4
Heavy Atoms 24
NP-Likeness -0.64

Activity Summary

IC50 2 meas. best 6.77

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.77 6.445 171.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
28246043 10.1016/j.ejmech.2017.02.040 Unchecked 2
28246043 10.1016/j.ejmech.2017.02.040 MDCK 1

Data from ChEMBL 36 via Core Engine