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Compound Detail

CHEMBL4170763

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Nc1nc(NC2CC2)c2nc[nH]c2n1

Basic Information

ChEMBL ID CHEMBL4170763
Phase Preclinical
Structure Type MOL
InChI Key IYWUSKBMXQERLH-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

190.2
MW (Da)
0.51
ALogP
5
HBA
3
HBD
92.5
PSA (Ų)
0.64
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C8H10N6
MW 190.21
Aromatic Rings 2
Heavy Atoms 14
NP-Likeness -0.95

Activity Summary

Kd 1 meas. best 4.6

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Kd 4.6 4.6 25000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked Kd = 25000.0 nM 4.6 Binding affinity to Clostridium difficile [5'-32P]guaA riboswitch by polyacrylam... 29220796

Literature References

PubMed DOI Target Context # Activities
29220796 10.1016/j.ejmech.2017.11.079 Clostridioides difficile 1
29220796 10.1016/j.ejmech.2017.11.079 Unchecked 1
29220796 10.1016/j.ejmech.2017.11.079 Escherichia coli 1

Data from ChEMBL 36 via Core Engine