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Compound Detail

CHEMBL417671

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O=C(Nc1ccccc1)c1ncn2c(=O)n(CCCl)nnc12

Basic Information

ChEMBL ID CHEMBL417671
Phase Preclinical
Structure Type MOL
InChI Key QODFDMULPJXWGM-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

318.7
MW (Da)
0.78
ALogP
7
HBA
1
HBD
94.2
PSA (Ų)
0.72
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H11ClN6O2
MW 318.72
Aromatic Rings 3
Heavy Atoms 22
NP-Likeness -1.95

Activity Summary

IC50 1 meas. best 5.9

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
TLX-5
CHEMBL615015
IC50 5.9 5.9 1250.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
TLX-5 IC50 = 1250.0 nM 5.9 In vitro cytotoxicity against mouse TLX5 lymphoma cells 7739008

Literature References

PubMed DOI Target Context # Activities
2329560 10.1021/jm00167a018 TLX-5 10
3806616 10.1021/jm00385a018 NON-PROTEIN TARGET 5
7739008 10.1021/jm00009a010 TLX-5 1

Data from ChEMBL 36 via Core Engine