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Compound Detail

CHEMBL440792

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C=C1[C@@H](CO)[C@H](O)C[C@H]1n1cnc2c(O)nc(N)nc21

Basic Information

ChEMBL ID CHEMBL440792
Phase Preclinical
Structure Type MOL
InChI Key QDGZDCVAUDNJFG-BWZBUEFSSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

277.3
MW (Da)
-0.42
ALogP
8
HBA
4
HBD
130.3
PSA (Ų)
0.55
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C12H15N5O3
MW 277.28
Aromatic Rings 2
Heavy Atoms 20
NP-Likeness 0.71

Activity Summary

EC50 1 meas. best 4.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
HepG2
CHEMBL395
EC50 4.0 4.0 100000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
HepG2 EC50 = 100000.0 nM 4.0 Tested for the effective concentration required to inhibit HBV in HepG2.2.15 hum... -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(96)00594-X HepG2 1

Data from ChEMBL 36 via Core Engine