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Compound Detail

CHEMBL44568

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CCCCCOC(=O)CC(CCn1cnc2c(O)nc(N)nc21)CC(=O)OCCCCC

Basic Information

ChEMBL ID CHEMBL44568
Phase Preclinical
Structure Type MOL
InChI Key OGLHAFOGJKOCRQ-UHFFFAOYSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

449.6
MW (Da)
3.37
ALogP
10
HBA
2
HBD
142.4
PSA (Ų)
0.31
QED
0
Ro5 Violations
15
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H35N5O5
MW 449.55
Aromatic Rings 2
Heavy Atoms 32
NP-Likeness -0.26

Activity Summary

IC50 2 meas. best 5.44

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vero
CHEMBL391
IC50 5.44 5.41 3600.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
3040998 10.1021/jm00392a020 Vero 2

Data from ChEMBL 36 via Core Engine