Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL4743948

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
Oc1ccc(CCNC(=S)Cc2ccc(O)c(O)c2)cc1O

Basic Information

ChEMBL ID CHEMBL4743948
Phase Preclinical
Structure Type MOL
InChI Key ADCANUVPVJYEKW-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

319.4
MW (Da)
2.21
ALogP
5
HBA
5
HBD
93.0
PSA (Ų)
0.43
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H17NO4S
MW 319.38
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness 0.09

Activity Summary

EC50 2 meas. best 5.89

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 5.89 5.89 1294.6 1
Influenza A virus
CHEMBL613740
EC50 5.15 5.15 7010.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
31954881 10.1016/j.ejmech.2020.112048 Unchecked 2
31954881 10.1016/j.ejmech.2020.112048 Influenza A virus 1
31954881 10.1016/j.ejmech.2020.112048 MDCK 1

Data from ChEMBL 36 via Core Engine