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Compound Detail

CHEMBL479529

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CCCCCCCCCCCCCCCCCCOCCOP(=O)([O-])CO[C@H](CO)Cn1ccc(N)nc1=O.[Na+]

Basic Information

ChEMBL ID CHEMBL479529
Phase Preclinical
Structure Type MOL
InChI Key AWNLXRBMSQEWNH-SNYZSRNZSA-M
Parent Compound CHEMBL206291
Active Moiety CHEMBL206291
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

575.7
MW (Da)
5.64
ALogP
9
HBA
3
HBD
146.1
PSA (Ų)
0.09
QED
2
Ro5 Violations
27
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H53N3NaO7P
MW 597.71
Aromatic Rings 1
Heavy Atoms 39
NP-Likeness 0.18

Activity Summary

IC50 2 meas. best 9.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Simplexvirus
CHEMBL613316
IC50 9.0 9.0 1.0 1
Vaccinia virus
CHEMBL613493
IC50 6.62 6.62 240.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Simplexvirus IC50 = 1.0 nM 9.0 Antiviral activity against Herpes simplex virus 19112024
Vaccinia virus IC50 = 240.0 nM 6.62 Antiviral activity against Vaccinia virus 19112024

Literature References

PubMed DOI Target Context # Activities
19112024 10.1016/j.bmc.2008.11.075 Vaccinia virus 1
19112024 10.1016/j.bmc.2008.11.075 Simplexvirus 1

Data from ChEMBL 36 via Core Engine