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Compound Detail

CHEMBL480863

METHYLINOSCAVIN B
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COc1cc(/C=C/c2cc3c(c(=O)o2)/C(=C/c2ccc(O)c(O)c2)C(C)(OC)O3)ccc1O

Basic Information

ChEMBL ID CHEMBL480863
Name METHYLINOSCAVIN B
Phase Preclinical
Structure Type MOL
InChI Key XCJITIROISCLRT-GAGKHWTPSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

450.4
MW (Da)
4.23
ALogP
8
HBA
3
HBD
118.6
PSA (Ų)
0.49
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C25H22O8
MW 450.44
Aromatic Rings 3
Heavy Atoms 33
NP-Likeness 1.51

Activity Summary

IC50 2 meas. best 4.88

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 4.88 4.65 13100.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
16499338 10.1021/np050453n NON-PROTEIN TARGET 2
16499338 10.1021/np050453n Radical scavenging activity 1

Data from ChEMBL 36 via Core Engine